Browse by Author

Temesszentandrasi-Ambrus, Csilla and Toth, Szilard and Verma, Rinkee and Banhegyi, Peter and Szabadkai, Istvan and Baska, Ferenc and Szantai-Kis, Csaba and Hartkoorn, Ruben C and Lingerfelt, Mary A and Sarkadi, Balazs and Szakacs, Gergely and Orfi, Laszlo and Nagaraja, Valakunja and Ekins, Sean and Telbisz, Agnes (2018) Characterization of new, efficient Mycobacterium tuberculosis topoisomerase-I inhibitors and their interaction with human ABC multidrug transporters. In: PLOS ONE, 13 (9).

Mori, Giorgia and Orena, Beatrice Silvia and Franch, Clara and Mitchenall, Lesley A and Godbole, Adwait Anand and Rodrigues, Liliana and Aguilar-Perez, Clara and Zemanova, Julia and Huszar, Stanislav and Forbak, Martin and Lane, Thomas R and Sabbah, Mohamad and Deboosere, Nathalie and Frita, Rosangela and Vandeputte, Alexandre and Hoffmann, Eik and Russo, Riccardo and Connel, Nancy and Veilleux, Courtney and Jha, Rajiv K and Kumar, Pradeep and Freundlich, Joel S and Brodin, Priscille and Ainsa, Jose Antonio and Nagaraja, Valakunja and Maxwell, Anthony and Mikusova, Katarina and Pasca, Maria Rosalia and Ekins, Sean (2018) The EU approved antimalarial pyronaridine shows antitubercular activity and synergy with rifampicin, targeting RNA polymerase. In: TUBERCULOSIS, 112 . pp. 98-109.

Ekins, Sean and Godbole, Adwait Anand and Keri, Gyorgy and Orfi, Laszlo and Pato, Janos and Bhat, Rajeshwari Subray and Verma, Rinkee and Bradley, Erin K and Nagaraja, Valakunja (2017) Machine learning and docking models for Mycobacterium tuberculosis topoisomerase I. In: TUBERCULOSIS, 103 . pp. 52-60.

Godbole, Adwait Anand and Ahmed, Wareed and Bhat, Rajeshwari Subray and Bradley, Erin K and Ekins, Sean and Nagaraja, Valakunja (2015) Targeting Mycobacterium tuberculosis Topoisomerase I by Small-Molecule Inhibitors. In: ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 59 (3). pp. 1554-1562.

Godbole, Adwait Anand and Ahmed, Wareed and Bhat, Rajeshwari Subray and Bradley, Erin K and Ekins, Sean and Nagaraja, Valakunja (2014) Inhibition of Mycobacterium tuberculosis topoisomerase I by m-AMSA, a eukaryotic type II topoisomerase poison. In: BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 446 (4). pp. 916-920.